Cypex - drug metabolism in vitro using recombinant cytochrome P450
Description
pulled from site's meta descriptionCypex - drug metabolism in vitro using recombinant cytochrome P450
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Categories:
- AboutUs AutoGen
- Cypex
- cypex
- Bactosomes
- bactosomes
- Bactosome
- bactosome
- cytochrome P450
- human cytochrome P450
- cytochrome P-450
- cytochrome+p450
- cytochrome+P450
- cytochrome+P-450
- cytochrome cyp
- cytochrome+cyp
- P450
- P-450
- p450
- CYP
- cyp
- EasyCYP
- drug metabolism
- inhibition
- CYP inhibition
- CYP+inhibition
- CYP inhibitor
- CYP+inhibitor
- p450 inhibition
- p450+inhibition
- P450 inhibition
- P450+inhibition
- p450 inhibition studies
- p450+inhibition+studies
- cyp inhibition studies
- cyp+inhibition+studies
- p450 inhibitor
- p450+inhibitor
- P450 inhibitor
- P450+inhibitor
- inhibition potential
- IC50
- Ki
- CYP+IC50
- p450+IC50
- direct inhibition
- direct+inhibition
- TDI
- time-dependent inhibition
- time-dependent+inhibition
- MDI
- metabolism-dependent inhibition
- metabolism-dependent+inhibition
- miconazole
- fluorometry
- fluorescence
- solvent
- in vitro
- in+vitro
- drug metabolising enzyme
- drug+metabolising+enzyme
- drug metabolizing enzyme
- drug+metabolizing+enzyme
- isoenzyme
- isozyme
- isoform
- reductase
- NADPH-cytochrome P450 reductase
- NADPH-CYP reductase
- NADPH P450-reductase
- P450-reductase
- CYP-reductase
- cytochrome b5
- b5
- metabolic profile
- metabolic profiling
- preclinical
- pre-clinical
- preclinical testing
- preclinical+testing
- pre-clinical testing
- pre-clinical+testing
- screening
- contract research
- CRO
- cro
- drug+metabolism
- drug development
- r&d
- R&D
- research
- development
- drug discovery
- ADME
- adme
- pharmacokinetic
- liver
- hepatic
- microsome
- substrate
- metabolite
- sulfotransferase
- sulphotransferase
- SULT
- glutathione S-transferase
- GST
- UDP-glucuronosyltransferase
- UDP-glucuronyltransferase
- UGT
- aldehyde oxidase
- aldehyde dehydrogenase
- carboxylesterase
- hCE1
- CES1
- hCE2
- CES2
- CYP1A1
- CYP1A2
- CYP1B1
- CYP1B1*1
- CYP1B1.1
- CYP1B1*3
- CYP1B1.3
- CYP1B1*4
- CYP1B1.4
- CYP2A6
- CYP2A13
- CYP2B6
- CYP2C8
- CYP2C9
- CYP2C9*1
- CYP2C9.1
- CYP2C9*2
- CYP2C9.2
- CYP2C9*3
- CYP2C9.3
- CYP2C18
- CYP2C19
- CYP2C20
- CYP2C43
- CYP2C75
- CYP2C76
- CYP2D6
- CYP2D6*1
- CYP2D6.1
- CYP2D6*2
- CYP2D6.2
- CYP2D6*10
- CYP2D6.10
- CYP2D6*39
- CYP2D6.39
- CYP2E1
- CYP2J2
- CYP3A4
- CYP3A5
- CYP3A7
- CYP3A8
- CYP4A11
- CYP4F2
- CYP4F3
- CYP4F3B
- CYP2B11
- CYP2C21
- CYP2C41
- CYP2D15
- CYP3A12
- CYP3A26
- Cyp2b10
- Cyp3a11
- beagle
- dog
- beagle dog
- canine
- cynomolgus
- monkey
- cynomolgus monkey
- mouse
- murine
- hydroxydiclofenac
- 4'-hydroxydiclofenac
- hydroxypaclitaxel
- lauric acid
- 14C lauric acid
- 14C+lauric acid
- 11-hydroxylauric acid
- 12-hydroxylauric acid
- tolbutamide
- hydroxytolbutamide
- carboxytolbutamide
- 7-ethoxyresorufin
- ethoxyresorufin
- 7ER
- resorufin
- 7-benzyloxyquinoline
- benzyloxyquinoline
- 7BQ
- 7-BQ
- 7bq
- 7-bq
- 7-hydroxyquinoline
- hydroxyquinoline
- 7HQ
- 7-HQ
- 7hq
- 7-hq
- 14C ethoxycoumarin
- 14C+ethoxycoumarin
- C14 ethoxycoumarin
- C14+ethoxycoumarin
- MAMC
- mamc
- HAMC
- hamc
- trifluoromethylcoumarin
- MFC
- mfc
- BFC
- bfc
- HFC
- hfc
- trifluoromethylumbelliferone
- omeprazole
- methylfluorescein
- 3-O-methylfluorescein
- OMF
- tienilic acid
- CYP2C9 inhibitor
- CYP2C9+inhibitor
- paclitaxel
- ketoconazole
- diclofenac
- amodiaquine
- desethylamodiaquine
- terfenadine
- N-benzylphenobarbital
- benzylphenobarbital
- NBPB
- CYP2C19 inhibitor
- CYP2C19+inhibitor
- montelukast
- diethoxyfluorescein
- DEF
- mephenytoin
- S-mephenytoin
- hydroxymephenytoin
- 4-hydroxymephenytoin
- 4'-hydroxymephenytoin
- SULT1A1
- SULT1A1*1
- SULT1A1.1
- SULT1A1*2
- SULT1A1.2
- SULT1A2
- SULT1A3
- SULT1B1
- SULT1C2
- SULT1C4
- SULT1E1
- SULT2A1
- GSTA1
- GSTM1
- UGT1A6
- antibody
- antibodies
- anti-cyp
- anti-CYP
- anti-p450
- anti-P450
- anti-SULT
- anti-SULT1A3
- polyclonal
- immunoinhibition
- immunoblotting
- Western blotting
- Western+blotting
- contract services
- reaction phenotyping
- reaction+phenotyping
- recombinant protein
- recombinant+protein
- protein expression
- protein+expression
- heterologous protein expression
- fermentation
- fermenter
- fermentor
- coli
- bacteria
- bacterial
- culture
- biotransformation
- biocatalysis
- metabolism
- metabolite synthesis
- metabolite+synthesis
- haem
- heme
- holoprotein
- purified cyp
- purified CYP
- purified p450
- purified p-450
- purified P450
- purified P-450